SCHEMBL9115585

SCHEMBL9115585

O=C1CCC(N2CCc3ccccc3C2)CC1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC18A3 Q16572 1/20 0.53
GRIN2B Q13224 3/20 0.46
CXCR3 P49682 1/20 0.46
MCOLN2 Q8IZK6 1/20 0.46
MCOLN3 Q8TDD5 1/20 0.46
MCOLN1 Q9GZU1 1/20 0.46
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
CRBN Q96SW2 1/20 0.44
KCNH2 Q12809 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
SMO Q99835 1/20 0.43
ADRA1A P35348 1/20 0.43
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
TMEM97 Q5BJF2 1/20 0.42
SIGMAR1 Q99720 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28286738 0.87 SLC18A3 (0.61) SLC18A3GRIN2BCXCR3MCOLN2MCOLN3
SCHEMBL8569045 0.84 GRIN2B (0.59) GRIN2BKCNH2HRH3
SCHEMBL10263767 0.84 SLC18A3 (0.67) SLC18A3GRIN2BCXCR3MCOLN2MCOLN3
SCHEMBL27781945 0.82 SLC18A3 (0.65) SLC18A3CXCR3MCOLN2MCOLN3MCOLN1
SCHEMBL8434677 0.81 MAOA (0.60) SLC18A3GRIN2BCXCR3MCOLN2MCOLN3
SCHEMBL30823779 0.80 SLC18A3 (0.50) SLC18A3GRIN2BCXCR3MCOLN2MCOLN3
SCHEMBL25833038 0.80 BRD4 (0.38) CXCR3CRBNKCNH2HRH3
SCHEMBL2299038 0.79 SLC18A3 (0.53) SLC18A3GRIN2BCXCR3MCOLN2MCOLN3
SCHEMBL29501341 0.79 SLC18A3 (0.53) SLC18A3CXCR3MAOAMAOBHRH3
SCHEMBL2657988 0.79 SLC18A3 (0.53) SLC18A3CXCR3MAOAMAOBHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995014469-A1 NOVEL SPIROCYCLES MERCK & CO., INC. (US) 1995-06-01 WO disclosed
US-5403846-A Antiarrhythmic agents MERCK & CO., INC. (US) 1995-04-04 US disclosed