SCHEMBL9115754

SCHEMBL9115754

CCCSC(N)=NCCC[C@H](N)C(=O)O

nearest known ligand 0.78

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 10/20 0.78
NOS2 P35228 9/20 0.78
NOS3 P29474 6/20 0.78
CYP2C19 P33261 3/20 0.68
THPO P40225 1/20 0.68
DDAH1 O94760 5/20 0.61
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
CYP1A2 P05177 2/20 0.58
TSHR P16473 2/20 0.58
GLA P06280 1/20 0.58
NFKB1 P19838 1/20 0.58
APEX1 P27695 1/20 0.58
CYP3A4 P08684 1/20 0.54
BLM P54132 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9141669 0.93 NOS1 (0.76) NOS1NOS2NOS3CYP2C19THPO
SCHEMBL9113062 0.91 NOS1 (0.74) NOS1NOS2NOS3CYP2C19THPO
SCHEMBL232480 0.88 NOS1 (1.00) NOS1NOS2NOS3CYP2C19THPO
SCHEMBL9141622 0.87 NOS2 (0.71) NOS1NOS2NOS3CYP2C19THPO
SCHEMBL29941582 0.83 NOS1 (0.74) NOS1NOS2NOS3CYP2C19THPO
SCHEMBL9114350 0.82 NOS1 (0.73) NOS1NOS2NOS3CYP2C19THPO
S-Methyl-D-Thiocitrulline SCHEMBL9114394 0.81 NOS1 (1.00) NOS1NOS2NOS3CYP2C19THPO
Thiocitrulline SCHEMBL940520 0.81 NOS1 (1.00) NOS1NOS2NOS3CYP2C19THPO
Thiocitrulline SCHEMBL4406617 0.80 NOS1 (0.97) NOS1NOS2NOS3CYP2C19THPO
Thiocitrulline SCHEMBL1320099 0.78 NOS2 (0.94) NOS1NOS2NOS3CYP2C19THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5476871-A Method for the treatment of hypotension induced by a cytokine or bacterial endotoxin using s-alkyl- isothioureido-amino acids THE MEDICAL COLLEGE OF WISCONSIN RESEARCH FOUNDATION, INC. (US) 1995-12-19 US disclosed
WO-1995013804-A1 S-ALKYL-ISOTHIOUREIDO-AMINO ACIDS AND USE THEREOF THE MEDICAL COLLEGE OF WISCONSIN RESEARCH FOUNDATION, INC. (US) 1995-05-26 WO disclosed
US-5364881-A S-alkyl-isothioureido-amino acids and use thereof THE MEDICAL COLLEGE OF WISCONSIN RESEARCH FOUNDATION, INC. (US) 1994-11-15 US disclosed