SCHEMBL9116434

SCHEMBL9116434

CS(=O)(=O)c1ccc(C2=CC3(C=C2c2ccc(C#N)cc2)CCC3)nc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.46
PTGS1 P23219 2/20 0.46
TNKS O95271 3/20 0.40
TNKS2 Q9H2K2 3/20 0.40
SULT2A1 Q06520 1/20 0.39
MLNR O43193 1/20 0.38
GPR119 Q8TDV5 1/20 0.37
CTSC P53634 1/20 0.36
LRRK2 Q5S007 3/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
ATR Q13535 1/20 0.35
CCR6 P51684 1/20 0.34
ALOX5AP P20292 1/20 0.34
KDM1A O60341 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117491 0.98 PTGS2 (0.46) PTGS2PTGS1TNKSTNKS2SULT2A1
SCHEMBL9117672 0.95 PTGS2 (0.51) PTGS2PTGS1TNKSTNKS2SULT2A1
SCHEMBL9117705 0.93 PTGS2 (0.49) PTGS2PTGS1GPR119LRRK2ATR
SCHEMBL9116918 0.89 CA2 (0.47) PTGS2PTGS1MLNRCA12CA1
SCHEMBL9116993 0.89 PTGS2 (0.54) PTGS2PTGS1GPR119LRRK2ATR
SCHEMBL9117586 0.87 CA2 (0.47) PTGS2PTGS1MLNRCA12CA1
SCHEMBL9117225 0.86 PTGS2 (0.50) PTGS2PTGS1GPR119ALOX5AP
SCHEMBL9118717 0.85 PTGS2 (0.49) PTGS2PTGS1ALOX5AP
SCHEMBL9117382 0.85 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL9118010 0.85 PTGS2 (0.48) PTGS2PTGS1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed