SCHEMBL9116473

SCHEMBL9116473

[C]1CCc2ccccc2OS1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
OXTR P30559 1/20 0.34
TSHR P16473 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.30
ITGB2 P05107 1/20 0.30
ICAM1 P05362 1/20 0.30
ITGAL P20701 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3995657 0.79 MAOA (0.38) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL29655819 0.72 MAOA (0.39) MAOAMAOBOXTRTSHRABCG2
SCHEMBL731982 0.72 MAOA (0.39) MAOAMAOBOXTRTSHRABCG2
SCHEMBL375376 0.72 MAOA (0.39) MAOAMAOBOXTRTSHRABCG2
SCHEMBL1724300 0.72 MAOA (0.39) MAOAMAOBOXTRTSHRABCG2
SCHEMBL4502914 0.69 TSHR (0.42) MAOAMAOBOXTRTSHRABCG2
SCHEMBL9119817 0.69 TSHR (0.42) MAOAMAOBOXTRTSHRABCG2
SCHEMBL124208 0.68 MAOA (0.39) MAOAMAOBOXTRTSHRABCG2
SCHEMBL654480 0.68 MAOA (0.35) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL1724509 0.67 MAOA (0.42) MAOAMAOBOXTRTSHRABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481920-B1 Benzoheterocyclylalkylaminoalkane diphosphonic acids CIBA GEIGY AG (CH) 1995-07-19 EP claimed
EP-0481920-A1 Benzoheterocyclylalkylaminoalkane diphosphonic acids CIBA-GEIGY AG (CH) 1992-04-22 EP claimed
EP-0423728-B1 Esters of castanospermine in the treatment of cerebral malaria MERRELL DOW PHARMA (US) 1995-08-30 EP disclosed
EP-0492841-B1 Anti-herpes castanospermine esters MERRELL DOW PHARMA (US) 1995-08-16 EP disclosed
EP-0481920-B1 Benzoheterocyclylalkylaminoalkane diphosphonic acids CIBA GEIGY AG (CH) 1995-07-19 EP disclosed
EP-0297534-B1 Castanospermine esters and glycosides MERRELL DOW PHARMA (US) 1994-12-28 EP disclosed
EP-0309952-B1 Anti-retroviral castanospermine esters MERRELL DOW PHARMA (US) 1994-06-22 EP disclosed
EP-0373663-B1 Castanospermine esters in the inhibition of tumor metastasis MERRELL DOW PHARMA (US) 1993-10-27 EP disclosed
EP-0492841-A1 Anti-herpes castanospermine esters MERRELL DOW PHARMACEUTICALS INC. (US) 1992-07-01 EP disclosed
EP-0481920-A1 Benzoheterocyclylalkylaminoalkane diphosphonic acids CIBA-GEIGY AG (CH) 1992-04-22 EP disclosed
US-5004746-A Anti-retroviral castanospermine esters MERRELL DOW PHARMACEUTICALS INC. (US) 1991-04-02 US disclosed
US-4952585-A Castanospermine esters in the inhibition of tumor metastasis MERRELL DOW PHARMACEUTICALS INC. (US) 1990-08-28 US disclosed