SCHEMBL9117643

SCHEMBL9117643

COc1ccc(-c2ccccc2)cc1-n1c(=O)[nH]c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.49
HSD17B10 Q99714 3/20 0.48
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
HPGD P15428 2/20 0.48
PKM P14618 1/20 0.47
HSP90AA1 P07900 5/20 0.47
HTR7 P34969 3/20 0.43
GABRP O00591 2/20 0.43
GABRD O14764 2/20 0.43
GABRA1 P14867 2/20 0.43
GABRB1 P18505 2/20 0.43
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
GABRA5 P31644 2/20 0.43
GABRA3 P34903 2/20 0.43
GABRA2 P47869 2/20 0.43
GABRB2 P47870 2/20 0.43
GABRA4 P48169 2/20 0.43
GABRE P78334 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118627 0.84 HSP90AA1 (0.54) PTPN1HSD17B10KDM4EALDH1A1HPGD
SCHEMBL9120265 0.83 HSP90AA1 (0.55) HSD17B10KDM4EALDH1A1HPGDPKM
SCHEMBL7479392 0.82 HTR7 (0.55) HSD17B10KDM4EALDH1A1HPGDPKM
SCHEMBL9119308 0.80 HSP90AA1 (0.72) KDM4EHSP90AA1GABRPGABRDGABRA1
SCHEMBL9117241 0.79 BCAT1 (0.41) PTPN1HSD17B10KDM4EALDH1A1HPGD
SCHEMBL30615640 0.76 ALDH1A1 (0.56) HSD17B10KDM4EALDH1A1HPGDPKM
SCHEMBL28904576 0.76 ALDH1A1 (0.56) HSD17B10KDM4EALDH1A1HPGDPKM
SCHEMBL4644935 0.76 PDE5A (0.52) HSD17B10KDM4EALDH1A1HPGDGABRP
SCHEMBL18934795 0.75 HSP90AA1 (0.52) KDM4EHPGDHSP90AA1GABRPGABRD
SCHEMBL5439923 0.73 HSP90AA1 (0.66) HPGDHSP90AA1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0477819-B1 Benzimidazole derivatives, their preparation and use NEUROSEARCH AS (DK) 1995-03-15 EP disclosed
US-5200422-A Benzimidazole derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-04-06 US disclosed
EP-0477819-A2 Benzimidazole derivatives, their preparation and use NEUROSEARCH A/S (DK) 1992-04-01 EP disclosed