SCHEMBL9119256

SCHEMBL9119256

NS(=O)(=O)c1ccc(C2=CC3(C=C2c2ccccc2)CCC3)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 9/20 0.40
CA1 P00915 8/20 0.40
CA9 Q16790 6/20 0.40
CA12 O43570 5/20 0.40
CA5A P35218 2/20 0.38
CA5B Q9Y2D0 2/20 0.38
CA4 P22748 1/20 0.38
FLT1 P17948 1/20 0.38
FLT4 P35916 1/20 0.38
KDR P35968 1/20 0.38
CA7 P43166 1/20 0.37
PTGS2 P35354 6/20 0.36
PTGS1 P23219 2/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
ALOX5AP P20292 2/20 0.35
IKBKB O14920 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9116102 0.97 CA2 (0.40) CA2CA1CA9CA12CA5A
SCHEMBL9117570 0.95 CA2 (0.41) CA2CA1CA9CA12CA5A
SCHEMBL9117334 0.88 PTGS2 (0.52) CA2CA1CA9CA5ACA5B
SCHEMBL9116501 0.88 PTGS2 (0.43) CA2CA1CA9CA12CA5A
SCHEMBL9116432 0.88 PTGS2 (0.43) CA2CA1CA9CA12CA5A
SCHEMBL9118010 0.88 PTGS2 (0.48) PTGS2PTGS1AKT1AKT2ALOX5AP
SCHEMBL9117988 0.85 PTGS2 (0.43) CA2CA1CA9CA12CA5A
SCHEMBL9239184 0.85 PTGS2 (0.43) CA2CA1CA9CA12CA5A
SCHEMBL9118428 0.85 PTGS2 (0.52) CA2CA1CA9CA5ACA5B
SCHEMBL9118085 0.85 PTGS2 (0.48) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed