SCHEMBL9124019

SCHEMBL9124019

O=[N+]([O-])c1cccc(C#Cc2ccccc2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.67
HSP90AA1 P07900 4/20 0.67
MAPT P10636 4/20 0.67
NPSR1 Q6W5P4 3/20 0.67
HTT P42858 3/20 0.67
OPRK1 P41145 2/20 0.67
S1PR2 O95136 1/20 0.67
FFAR1 O14842 1/20 0.64
KMT2A Q03164 4/20 0.62
MEN1 O00255 3/20 0.62
SMN1; SMN2 Q16637 2/20 0.62
MITF O75030 1/20 0.62
TSHR P16473 3/20 0.59
LMNA P02545 2/20 0.59
NFE2L2 Q16236 1/20 0.53
ACHE P22303 1/20 0.50
TP53 P04637 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ALOX15 P16050 1/20 0.50
CASP3 P42574 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28728423 0.94 TSHR (0.67) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL18561137 0.86 VCAM1 (0.53) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL13717179 0.86 ALDH1A1 (0.52) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL18561131 0.85 FFAR1 (0.52) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL13622489 0.84 ALDH1A1 (0.70) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL29433452 0.83 TSHR (0.57) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL3874391 0.83 ALDH1A1 (0.60) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL1507602 0.83 TSHR (0.57) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL10729521 0.83 TSHR (0.57) ALDH1A1HSP90AA1MAPTNPSR1HTT
SCHEMBL12350152 0.82 NFE2L2 (0.57) ALDH1A1HSP90AA1MAPTNPSR1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248455-A 3, 5-disubstituted isoxazole derivatives and synthesis method thereof 湖北科技学院 2021-08-13 CN claimed
EP-0443352-B1 Polyimides end-capped with diaryl substituted acetylene NAT STARCH CHEM INVEST (US) 1995-12-06 EP disclosed
US-5449740-A Resin systems derived from insitu-generated bisdienes from bis-benzocyclobutene compounds THE UNIVERSITY OF DAYTON (US) 1995-09-12 US disclosed
US-5138028-A Composites, molding materials, adhesives, electronics NATIONAL STARCH AND CHEMICAL INVESTMENT HOLDING CORPORATION (US) 1992-08-11 US disclosed
EP-0443352-A2 Polyimides end-capped with diaryl substituted acetylene National Starch and Chemical Investment Holding Corporation (US) 1991-08-28 EP disclosed
EP-0001479-A2 Process for the preparation of nitrophenylhydroxyacetylene and conversion to nitrophenylacetylene GULF RESEARCH & DEVELOPMENT COMPANY (US) 1979-04-18 EP disclosed
US-4128588-A PALLADIUM-PHOSPHINE COMPLEX CATALYST GULF RESEARCH & DEVELOPMENT COMPANY (US) 1978-12-05 US disclosed