SCHEMBL9125643

SCHEMBL9125643

N#Cc1ccc(NC(=S)Nc2ncccc2OCc2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPIA P62937 15/20 0.60
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C19 P33261 1/20 0.53
ALDH1A1 P00352 2/20 0.52
RECQL P46063 1/20 0.52
PPIF P30405 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9125099 0.88 PPIA (0.72) PPIAMEN1KMT2ACYP1A2CYP2C19
SCHEMBL9125711 0.87 PPIA (0.60) PPIAPPIF
SCHEMBL9126145 0.85 PPIA (0.75) PPIAMEN1KMT2ACYP1A2CYP2C19
SCHEMBL9124984 0.82 PPIA (0.77) PPIAMEN1KMT2ACYP1A2CYP2C19
SCHEMBL9124394 0.81 PPIA (0.68) PPIAMEN1KMT2ACYP1A2CYP2C19
SCHEMBL9126266 0.80 MEN1 (0.61) PPIAMEN1KMT2AALDH1A1
SCHEMBL9125557 0.80 PPIA (0.60) PPIAMEN1KMT2ACYP1A2CYP2C19
SCHEMBL9125727 0.78 PPIA (0.56) PPIAPPIF
SCHEMBL2335868 0.76 PPIA (0.64) PPIAPPIF
SCHEMBL9125484 0.76 PPIA (0.61) PPIAMEN1KMT2AALDH1A1PPIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed