SCHEMBL9125727

SCHEMBL9125727

N#Cc1ccc(N=C(N)Nc2ncccc2OCc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPIA P62937 16/20 0.56
MAOB P27338 1/20 0.44
PPIF P30405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2783284 0.89 PPIA (0.58) PPIAPPIF
SCHEMBL9125077 0.86 PPIA (0.62) PPIAPPIF
SCHEMBL9126116 0.83 PPIA (0.64) PPIAPPIF
SCHEMBL9125087 0.81 PPIA (0.59) PPIAPPIF
SCHEMBL9127376 0.81 PPIA (0.53) PPIAPPIF
SCHEMBL9128504 0.81 NPC1 (0.54) PPIA
SCHEMBL9125711 0.78 PPIA (0.60) PPIAMAOBPPIF
SCHEMBL9125643 0.78 PPIA (0.60) PPIAPPIF
SCHEMBL9122341 0.77 PPIA (0.51) PPIAPPIF
SCHEMBL9124791 0.76 NPC1 (0.51) PPIAPPIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed