SCHEMBL9129696

SCHEMBL9129696

CN(C)c1ccc(C(=O)C#Cc2cccs2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.54
ALDH1A1 P00352 3/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 2/20 0.43
RAB9A P51151 4/20 0.42
NPC1 O15118 4/20 0.42
KMT2A Q03164 4/20 0.39
CASP3 P42574 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP1B1 Q16678 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
POLB P06746 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
VCP P55072 1/20 0.39
JAK3 P52333 1/20 0.38
GFER P55789 1/20 0.37
MEN1 O00255 3/20 0.37
KDM4E B2RXH2 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7201310 0.83 VCP (0.57) ALDH1A1MAPTHPGDRAB9ANPC1
SCHEMBL7200606 0.81 APP (0.49) APPALDH1A1MAPTHPGDRAB9A
SCHEMBL7202747 0.81 HSP90AA1 (0.49) ALDH1A1MAPTHPGDRAB9ANPC1
SCHEMBL7204230 0.80 APP (0.47) APPALDH1A1MAPTRAB9ANPC1
SCHEMBL7204585 0.80 APP (0.51) APPALDH1A1MAPTHPGDRAB9A
SCHEMBL7203532 0.80 MAPT (0.44) MAPTKMT2ASMN1; SMN2CYP1B1POLB
SCHEMBL7203523 0.80 RAB9A (0.49) ALDH1A1MAPTHPGDRAB9ANPC1
SCHEMBL7200084 0.79 RAB9A (0.50) ALDH1A1MAPTHPGDRAB9ANPC1
SCHEMBL7202454 0.79 MAPT (0.46) ALDH1A1MAPTRAB9ANPC1KMT2A
SCHEMBL7200878 0.79 APP (0.54) APPALDH1A1MAPTHPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0476645-B1 Calcium uptake inhibitors MERRELL DOW PHARMA (US) 1995-09-06 EP disclosed
US-5409942-A Administering 1-phenyl-3-aryl-2-propyne-1-ones compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-25 US disclosed
US-5223518-A Controlling intake in leukocytes and platelets MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-29 US disclosed
EP-0476645-A1 Calcium uptake inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1992-03-25 EP disclosed