SCHEMBL9130467

SCHEMBL9130467

CN(C)c1ccc(C(O)C#C[Si](C)(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.40
TSHR P16473 3/20 0.39
HSD17B10 Q99714 2/20 0.39
ALOX15 P16050 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 4/20 0.38
ATM Q13315 1/20 0.38
MAPT P10636 2/20 0.38
POLB P06746 1/20 0.38
FFAR1 O14842 1/20 0.37
SLC2A1 P11166 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KDM4E B2RXH2 2/20 0.36
CACNA2D1 P54289 1/20 0.36
CACNB2 Q08289 1/20 0.36
CACNA1C Q13936 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9547906 0.85 ALDH1A1 (0.50) ALDH1A1TSHRHSD17B10ALOX15MEN1
SCHEMBL9133521 0.81 ALDH1A1 (0.44) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL2800138 0.78 ALOX5 (0.40) ALDH1A1KMT2AATMPOLBFFAR1
SCHEMBL2799259 0.77 CACNA2D1 (0.56) ALDH1A1TSHRHSD17B10ALOX15MEN1
SCHEMBL8013623 0.76 ALDH1A1 (0.44) ALDH1A1TSHRHSD17B10MEN1KMT2A
SCHEMBL14677386 0.76 CACNA2D1 (0.39) ALDH1A1HSD17B10MEN1KMT2AGAA
SCHEMBL2197891 0.75 ALOX5 (0.46) KDM4ECACNA2D1CACNB2CACNA1C
SCHEMBL9131675 0.75 CHRM5 (0.47) ALDH1A1TSHRHSD17B10ALOX15MEN1
SCHEMBL6971747 0.73 ALDH1A1 (0.46) ALDH1A1TSHRHSD17B10ALOX15MEN1
SCHEMBL1578958 0.73 TSHR (0.54) ALDH1A1TSHRHSD17B10ALOX15MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0476645-B1 Calcium uptake inhibitors MERRELL DOW PHARMA (US) 1995-09-06 EP disclosed
US-5409942-A Administering 1-phenyl-3-aryl-2-propyne-1-ones compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-25 US disclosed
US-5223518-A Controlling intake in leukocytes and platelets MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-29 US disclosed
EP-0476645-A1 Calcium uptake inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1992-03-25 EP disclosed