SCHEMBL9130737

SCHEMBL9130737

COC(=O)c1ccc2cc(-c3ccc(C(C)(C)C)cc3)sc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.56
HDAC6 Q9UBN7 5/20 0.52
HDAC3 O15379 2/20 0.50
HDAC2 Q92769 2/20 0.50
HDAC8 Q9BY41 2/20 0.50
NPSR1 Q6W5P4 5/20 0.48
MAPK1 P28482 2/20 0.48
KDM4E B2RXH2 4/20 0.47
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CRHBP P24387 2/20 0.46
CRHR2 Q13324 2/20 0.46
GFER P55789 1/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
EGFR P00533 1/20 0.44
KIF11 P52732 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8459958 0.85 HDAC6 (0.50) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL498889 0.85 ESR1 (0.60) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL497643 0.84 HDAC6 (0.62) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL9133624 0.77 HDAC1 (0.51) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL732990 0.77 APP (0.58) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL3144561 0.76 ESR1 (0.73) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL1886145 0.76 HDAC1 (0.80) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL13008716 0.75 CA1 (0.62) HDAC1MAPK1CA1CA2EGFR
SCHEMBL19029168 0.74 HDAC6 (0.70) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL263634 0.74 KIF11 (0.57) HDAC1NPSR1MAPK1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428052-A Classifiable as retinoids; skin disorders, corneopathy CENTRE INTERNATIONALE DE RECHERCHES DERMATOLOGIQUES (C.I.R.D.) (FR) 1995-06-27 US disclosed
US-5288744-A Tetramethyltetrahydronaphthyl benzothiazole for treating skin disorders CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (C.I.R.D.) (FR) 1994-02-22 US disclosed
US-5260295-A Retinoic acid derivatives, cosmetics, skin disorders CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (C.I.R.D.) (FR) 1993-11-09 US disclosed
US-5059621-A Treatment of dermatologic ailments linked to keratinization disorder CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (C.I.R.D.) (FR) 1991-10-22 US disclosed
US-4920140-A Skin disorders CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES C.I.R.D. (FR) 1990-04-24 US disclosed
US-4740519-A Benzo (b) thiophene carboxylate derivatives and pharmaceutical compositions CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES C.I.R.D. (FR) 1988-04-26 US disclosed