SCHEMBL9130762

SCHEMBL9130762

N#Cc1ccccc1Oc1ccccc1NC(=O)c1ccc(OCc2ccc3ccccc3n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.54
CYSLTR1 Q9Y271 7/20 0.48
PDE10A Q9Y233 3/20 0.48
CYSLTR2 Q9NS75 2/20 0.47
MAPK14 Q16539 1/20 0.46
FFAR1 O14842 1/20 0.46
AKR1B1 P15121 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9131337 0.85 GPBAR1 (0.53) GPBAR1CYSLTR1PDE10ACYSLTR2FFAR1
SCHEMBL9132216 0.79 CACNA1H (0.53) MAPK14
SCHEMBL9131506 0.79 GPBAR1 (0.49) GPBAR1CYSLTR1PDE10ACYSLTR2
SCHEMBL9129427 0.79 PLK1 (0.61) MAPK14
SCHEMBL9130582 0.78 CACNA1H (0.54) MAPK14
SCHEMBL9135886 0.76 ALDH1A1 (0.43) GPBAR1CYSLTR1CYSLTR2
SCHEMBL9132696 0.76 CACNA1H (0.52) MAPK14
SCHEMBL3534448 0.76 GPBAR1 (0.74) GPBAR1CYSLTR1PDE10ACYSLTR2FFAR1
SCHEMBL9130515 0.76 LMNA (0.58) MAPK14
SCHEMBL10663836 0.75 CYSLTR1 (0.56) GPBAR1CYSLTR1PDE10ACYSLTR2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5399703-A Antiallergens NIPPON SHINYAKU COMPANY, LIMITED (JP) 1995-03-21 US disclosed
EP-0536400-A1 TETRAZOLE DERIVATIVE AND MEDICINE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-04-14 EP disclosed