SCHEMBL9132015

SCHEMBL9132015

CC(C)NCCCOc1ccccc1C(=O)Nc1cccc2[nH]ccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 3/20 0.60
HTR1A P08908 5/20 0.49
HDAC3 O15379 1/20 0.47
BRD4 O60885 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
NR2E1 Q9Y466 1/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
LMNA P02545 2/20 0.46
ADRB2 P07550 2/20 0.46
ADRB1 P08588 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9130186 0.92 HTR1B (0.60) HTR1BHTR1AHDAC3BRD4HDAC4
SCHEMBL9132886 0.86 HTR1A (0.48) HTR1BHTR1AHDAC3BRD4HDAC4
SCHEMBL9130336 0.86 DHPS (0.50) HTR1BHDAC3BRD4HDAC4HDAC1
SCHEMBL9130728 0.85 HDAC3 (0.52) HDAC3BRD4HDAC4HDAC1HDAC7
SCHEMBL9133428 0.85 DHPS (0.51) HTR1BHDAC3BRD4HDAC4HDAC1
SCHEMBL9133110 0.84 HTR1A (0.69) HTR1BHTR1ANR2E1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9739316 0.84 DHPS (0.50) HTR1BHDAC3BRD4HDAC4HDAC1
SCHEMBL9132132 0.84 RXFP1 (0.46) HTR1BHTR1AHDAC3BRD4HDAC4
SCHEMBL9136237 0.83 DHPS (0.47) HTR1BHDAC3BRD4HDAC4HDAC1
SCHEMBL9131204 0.83 DHPS (0.47) HTR1BHDAC3BRD4HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380722-A Antiarrhythmia agents ROUSSEL-UCLAF (FR) 1995-01-10 US disclosed