SCHEMBL9149795

SCHEMBL9149795

COc1ccc2sc(C3CCCC(C)C3)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.46
CA2 P00918 1/20 0.41
HTR1A P08908 2/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
CLK1 P49759 9/20 0.39
DYRK1A Q13627 4/20 0.39
DYRK1B Q9Y463 1/20 0.39
TSHR P16473 1/20 0.38
CHRNA7 P36544 2/20 0.36
CLK2 P49760 3/20 0.36
CLK4 Q9HAZ1 1/20 0.36
HTR3A P46098 1/20 0.35
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8601033 0.90 HTR1A (0.41) CA2HTR1ATSHRCHRNA7SLC6A4
SCHEMBL9151822 0.86 BACE1 (0.53) BACE1CA2HTR1APDE3BPDE3A
SCHEMBL4450281 0.76 CA2 (0.48) BACE1CA2HTR1ACHRNA7SLC6A4
SCHEMBL4442733 0.75 CA2 (0.47) BACE1CA2HTR1ADYRK1ACHRNA7
SCHEMBL4442739 0.75 CA2 (0.47) BACE1CA2HTR1ADYRK1ACHRNA7
SCHEMBL8601229 0.75 CA2 (0.47) BACE1CA2HTR1ADYRK1ACHRNA7
SCHEMBL4438841 0.75 CA2 (0.47) BACE1CA2HTR1ADYRK1ACHRNA7
SCHEMBL4442755 0.75 CA2 (0.47) BACE1CA2HTR1ADYRK1ACHRNA7
SCHEMBL4444144 0.73 CA2 (0.46) BACE1CA2HTR1APDE3BPDE3A
SCHEMBL5756786 0.70 HTR1A (0.43) CA2HTR1APDE3BPDE3ACHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5472962-A Antiestrogenic agents TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-12-05 US disclosed
US-5449812-A Substituted benzenesulfonamide derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1995-09-12 US disclosed