SCHEMBL9150250

SCHEMBL9150250

Cc1ccc2c(C3CCN(CCN4CCNC4=O)CC3)c[nH]c2c1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.53
SLC6A4 P31645 1/20 0.53
ADRA1D P25100 2/20 0.48
HTR2A P28223 2/20 0.48
KCNH2 Q12809 3/20 0.47
HTR7 P34969 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9372780 0.87 KCNH2 (0.61) DRD2SLC6A4ADRA1DHTR2AKCNH2
SCHEMBL9150449 0.82 DRD2 (0.49) DRD2SLC6A4ADRA1DHTR2AKCNH2
SCHEMBL23010845 0.78 APP (0.64) DRD2SLC6A4ADRA1D
SCHEMBL9149801 0.75 KCNH2 (0.61) DRD2SLC6A4ADRA1DHTR2AKCNH2
SCHEMBL6958224 0.75 HTR1A (0.66) DRD2
SCHEMBL9153282 0.75 KCNH2 (0.77) DRD2SLC6A4ADRA1DHTR2AKCNH2
SCHEMBL8642590 0.73 HTR1A (0.80) DRD2SLC6A4ADRA1DHTR2AKCNH2
SCHEMBL18324794 0.72 IDO1 (0.47) DRD2SLC6A4ADRA1DHTR2AKCNH2
SCHEMBL4676883 0.72 HTR2C (0.62) DRD2SLC6A4HTR2A
SCHEMBL9153185 0.72 ADRA1D (0.52) SLC6A4ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5457115-A Treating anxiety, depression, sleep disorders, migranes, schizophrenia or Parkinson's disease in humans H. LUNDBECK A/S (DK) 1995-10-10 US disclosed
EP-0465398-B1 Novel indole derivatives LUNDBECK & CO AS H (DK) 1994-12-14 EP disclosed
US-5322851-A Indole derivatives H. LUNDBECK A/S (DK) 1994-06-21 US disclosed
US-5216001-A Central nervous system disorders H. LUNBECK A/S (DK) 1993-06-01 US disclosed
EP-0465398-A2 Novel indole derivatives H. LUNDBECK A/S (DK) 1992-01-08 EP disclosed