SCHEMBL9150307

SCHEMBL9150307

Cc1cc2ccccc2n1-c1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.48
NOTUM Q6P988 1/20 0.45
GRIA1 P42261 1/20 0.43
CACNG8 Q8WXS5 1/20 0.43
CACNG2 Q9Y698 1/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
TSHR P16473 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HKDC1 Q2TB90 2/20 0.41
MAPK1 P28482 1/20 0.39
SCN9A Q15858 2/20 0.39
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13425012 0.91 ALDH1A1 (0.47) CYP19A1NOTUMKDM4EALDH1A1KMT2A
SCHEMBL12345965 0.85 ALDH1A1 (0.43) CYP19A1NOTUMGRIA1CACNG8CACNG2
SCHEMBL30446730 0.85 ALDH1A1 (0.55) CYP19A1NOTUMKDM4EALDH1A1KMT2A
SCHEMBL1885602 0.85 ALDH1A1 (0.55) CYP19A1NOTUMKDM4EALDH1A1KMT2A
SCHEMBL13483671 0.83 TSHR (0.43) CYP19A1NOTUMKDM4EALDH1A1KMT2A
SCHEMBL76833 0.82 ESR2 (0.47) CYP19A1NOTUMGRIA1CACNG8CACNG2
SCHEMBL6986420 0.82 ALDH1A1 (0.44) CYP19A1KDM4EALDH1A1KMT2AMEN1
SCHEMBL13241999 0.82 APP (0.46) CYP19A1NOTUMKDM4EALDH1A1KMT2A
SCHEMBL9267750 0.81 POLB (0.46) CYP19A1NOTUMKDM4EKMT2AMEN1
SCHEMBL64405 0.79 ALDH1A1 (0.44) NOTUMKDM4EALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5457115-A Treating anxiety, depression, sleep disorders, migranes, schizophrenia or Parkinson's disease in humans H. LUNDBECK A/S (DK) 1995-10-10 US disclosed
EP-0465398-B1 Novel indole derivatives LUNDBECK & CO AS H (DK) 1994-12-14 EP disclosed
US-5322851-A Indole derivatives H. LUNDBECK A/S (DK) 1994-06-21 US disclosed
US-5216001-A Central nervous system disorders H. LUNBECK A/S (DK) 1993-06-01 US disclosed