SCHEMBL9154232

SCHEMBL9154232

COc1ccc(CN2CCN(C(=O)[C@@H](N)Cc3ccccc3)CC2)c(OC)c1OC

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.60
HTT P42858 1/20 0.60
CYP2C19 P33261 1/20 0.59
KDM4E B2RXH2 6/20 0.58
PKM P14618 1/20 0.58
MEN1 O00255 8/20 0.57
KMT2A Q03164 8/20 0.57
RECQL P46063 1/20 0.51
ALOX15 P16050 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
GAA P10253 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CYP1A2 P05177 1/20 0.48
CHRM2 P08172 1/20 0.48
SLC6A4 P31645 1/20 0.48
OPRD1 P41143 1/20 0.48
OPRK1 P41145 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9426502 0.99 ALDH1A1 (0.59) ALDH1A1HTTCYP2C19KDM4EPKM
SCHEMBL9154459 0.87 ALDH1A1 (0.56) ALDH1A1HTTCYP2C19KDM4EPKM
SCHEMBL9154894 0.85 CYP2C19 (0.61) ALDH1A1HTTCYP2C19KDM4EPKM
SCHEMBL9426259 0.84 CYP2C19 (0.60) ALDH1A1HTTCYP2C19KDM4EPKM
SCHEMBL10858976 0.84 CYP2C19 (0.69) ALDH1A1HTTCYP2C19KDM4EPKM
SCHEMBL10858979 0.84 CYP2C19 (0.69) ALDH1A1HTTCYP2C19KDM4EPKM
SCHEMBL9158845 0.83 CYP2C19 (0.71) ALDH1A1HTTCYP2C19KDM4EPKM
SCHEMBL9160121 0.83 CYP2C19 (0.71) ALDH1A1HTTCYP2C19KDM4EPKM
Hydrochloric Acid SCHEMBL10859968 0.83 CYP2C19 (0.67) ALDH1A1HTTCYP2C19KDM4EPKM
Hydrochloric Acid SCHEMBL10859963 0.83 CYP2C19 (0.67) ALDH1A1HTTCYP2C19KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533516-B1 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-02-08 EP disclosed
US-5340809-A Antihypoxic, antiischemic agents ADIR ET COMPAGNIE (FR) 1994-08-23 US disclosed
EP-0533516-A2 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-03-24 EP disclosed