SCHEMBL9154459

SCHEMBL9154459

COc1ccc(CN2CCN(C(=O)[C@@H](N)CSCc3ccccc3)CC2)c(OC)c1OC

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.56
HTT P42858 1/20 0.56
CYP2C19 P33261 1/20 0.54
MEN1 O00255 9/20 0.53
KMT2A Q03164 9/20 0.53
KDM4E B2RXH2 6/20 0.51
PKM P14618 1/20 0.51
RECQL P46063 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
ALOX15 P16050 1/20 0.46
GAA P10253 1/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9154232 0.87 ALDH1A1 (0.60) ALDH1A1HTTCYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL9426502 0.86 ALDH1A1 (0.59) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9425650 0.86 NPC1 (0.54) ALDH1A1MEN1KMT2AKDM4ERECQL
SCHEMBL9425638 0.85 ALDH1A1 (0.55) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9426122 0.84 ALDH1A1 (0.53) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9154438 0.83 ALDH1A1 (0.51) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9425617 0.83 ALDH1A1 (0.51) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9158912 0.82 CYP2C19 (0.58) ALDH1A1HTTCYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL9425757 0.82 ALDH1A1 (0.51) ALDH1A1HTTCYP2C19MEN1KMT2A
SCHEMBL9154894 0.81 CYP2C19 (0.61) ALDH1A1HTTCYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533516-B1 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-02-08 EP claimed
EP-0533516-A2 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-03-24 EP claimed