SCHEMBL9155290

SCHEMBL9155290

O=[N+]([O-])c1ccccc1N1CCN(CCCl)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.58
HTT P42858 2/20 0.56
KMT2A Q03164 1/20 0.56
DRD2 P14416 4/20 0.55
HTR2A P28223 3/20 0.55
HTR7 P34969 3/20 0.55
HTR6 P50406 3/20 0.55
MITF O75030 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
MAPT P10636 1/20 0.53
MAPK1 P28482 1/20 0.53
CCR6 P51684 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
DRD4 P21917 2/20 0.53
DRD3 P35462 1/20 0.53
ENPP2 Q13822 2/20 0.49
GRM5 P41594 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23536279 0.85 HTR1A (0.58) HTR1AHTTKMT2ADRD2HTR2A
SCHEMBL29932017 0.85 HTR1A (0.58) HTR1AHTTKMT2ADRD2HTR2A
Hydrochloric Acid SCHEMBL31232826 0.84 HTR1A (0.57) HTR1AHTTKMT2ADRD2HTR2A
SCHEMBL1274938 0.84 HTT (0.73) HTR1AHTTKMT2AMITFALDH1A1
SCHEMBL8828404 0.83 DRD2 (0.59) HTR1AHTTKMT2ADRD2HTR2A
SCHEMBL27351820 0.83 DRD2 (0.58) HTR1AHTTKMT2ADRD2HTR2A
SCHEMBL4520581 0.82 KMT2A (0.61) HTR1AHTTKMT2ADRD2MITF
SCHEMBL24629113 0.82 HTR1A (0.58) HTR1AHTTKMT2ADRD2HTR2A
SCHEMBL3210395 0.82 DRD2 (0.60) HTR1AHTTKMT2ADRD2HTR2A
SCHEMBL18118448 0.82 DRD2 (0.58) HTR1AHTTKMT2ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405847-A Antiallergic, antiasthmatic, anxiolytic, hypotensive agents ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1995-04-11 US disclosed
EP-0584487-A2 4,5-Dihydro-4-oxopyrrolo (1,2-a) quinoxalines and aza-analoges and process for their preparation ASTA Medica Aktiengesellschaft (DE) 1994-03-02 EP disclosed