SCHEMBL8828404

SCHEMBL8828404

O=[N+]([O-])c1ccccc1N1CCN(CCCO)CC1

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.59
DRD4 P21917 2/20 0.59
DRD3 P35462 1/20 0.59
HTR1A P08908 4/20 0.58
HTR7 P34969 4/20 0.58
HTR2A P28223 3/20 0.58
HTR6 P50406 3/20 0.58
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
HTT P42858 1/20 0.53
KMT2A Q03164 1/20 0.53
MAPK1 P28482 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27351820 0.86 DRD2 (0.58) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL9612238 0.85 DRD2 (0.62) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL3210388 0.85 DRD2 (0.59) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL3210395 0.85 DRD2 (0.60) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL3482338 0.84 SIGMAR1 (0.72) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL23536279 0.83 HTR1A (0.58) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL9155290 0.83 HTR1A (0.58) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL29932017 0.83 HTR1A (0.58) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL18118448 0.82 DRD2 (0.58) DRD2DRD4DRD3HTR1AHTR7
Hydrochloric Acid SCHEMBL31232826 0.82 HTR1A (0.57) DRD2DRD4DRD3HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
CN-1136039-A [3- (4-phenylpiperazin-1-yl) propylamino, thio and oxy ] -pyridine, pyrimidine and benzene derivatives HOFFMANN LA ROCHE (CH) 1996-11-20 CN disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed