SCHEMBL9155804

SCHEMBL9155804

CC(C)(C=O)Cc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.48
TSHR P16473 2/20 0.46
IDO1 P14902 2/20 0.44
ALDH1A1 P00352 4/20 0.44
ACHE P22303 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CHRM2 P08172 1/20 0.44
CYP2C19 P33261 3/20 0.43
POLB P06746 1/20 0.43
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
CYP1A2 P05177 3/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPK1 P28482 1/20 0.41
BLM P54132 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL75530 0.81 LOXL2 (0.55) LOXL2TSHRIDO1ALDH1A1ACHE
SCHEMBL9163048 0.80 TSHR (0.54) TSHRALDH1A1ACHECYP2C19POLB
SCHEMBL1627332 0.78 TSHR (0.53) LOXL2TSHRIDO1ALDH1A1ACHE
SCHEMBL776520 0.78 LOXL2 (0.57) LOXL2TSHRIDO1ALDH1A1ACHE
SCHEMBL7107843 0.78 LOXL2 (0.52) LOXL2TSHRIDO1ALDH1A1ACHE
SCHEMBL97944 0.78 LOXL2 (0.52) LOXL2TSHRIDO1ALDH1A1ACHE
SCHEMBL7107845 0.76 LOXL2 (0.50) LOXL2TSHRIDO1ALDH1A1ACHE
SCHEMBL18387787 0.76 TSHR (0.52) LOXL2TSHRIDO1ALDH1A1ACHE
SCHEMBL18387801 0.76 LOXL2 (0.50) LOXL2TSHRIDO1ALDH1A1ACHE
SCHEMBL9307922 0.75 LOXL2 (0.58) LOXL2TSHRIDO1ALDH1A1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1040753-C Pyridine derivatives and the preparation thereof ICI PLC (GB) 1998-11-18 CN disclosed
US-5401849-A FOR ANTAGONIZING THE ACTIONS OF, AND INHIBITING THE SYNTHESIS OF, THROMBOXANE A2 ZENECA LIMITED (GB) 1995-03-28 US disclosed
EP-0329360-B1 Pyridine derivatives ICI PLC (GB) 1994-08-03 EP disclosed
US-5248780-A Thromboxane inhibitors IMPERIAL CHEMICAL INDUSTRIES, PLC (GB) 1993-09-28 US disclosed
US-5166213-A Antiischemic agents, cardiovascular disorders, antiasthmatics or antiinflammatory agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-11-24 US disclosed
CN-1035115-A Pyridine derivate and preparation method thereof ICI PLC (GB) 1989-08-30 CN disclosed
EP-0329360-A2 Pyridine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-08-23 EP disclosed