SCHEMBL9158940

SCHEMBL9158940

CCCCCCC1CCC(C(C)c2ccc(-c3ccc(F)nc3)cc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
PTGS2 P35354 1/20 0.34
APLNR P35414 6/20 0.34
GRIA2 P42262 5/20 0.33
KCNH2 Q12809 3/20 0.33
GBA1 P04062 1/20 0.32
UGCG Q16739 1/20 0.32
GBA2 Q9HCG7 1/20 0.32
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
MMP13 P45452 1/20 0.31
TP53 P04637 1/20 0.31
CYP2E1 P05181 1/20 0.31
CYP2A6 P11509 1/20 0.31
CYP2B6 P20813 1/20 0.31
ACACB O00763 1/20 0.31
ACACA Q13085 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9156816 1.00 GAA (0.35) GAAMAPTPTGS2APLNRGRIA2
SCHEMBL9157491 0.99 PTGS2 (0.35) GAAMAPTPTGS2APLNRGRIA2
SCHEMBL9155759 0.95 PTGS2 (0.35) GAAPTGS2APLNRGRIA2KCNH2
SCHEMBL9158474 0.90 PTGS2 (0.36) PTGS2APLNRGRIA2KCNH2MMP2
SCHEMBL9154581 0.86 PSEN1 (0.38) GAAMAPTPTGS2
SCHEMBL9158482 0.86 PSEN1 (0.38) GAAMAPTPTGS2
SCHEMBL9157702 0.86 GAA (0.35) GAAMAPTTP53CYP2A6ACACB
SCHEMBL9160035 0.86 GAA (0.35) GAAMAPTTP53CYP2A6ACACB
SCHEMBL8774654 0.85 GAA (0.33) GAAMAPTPTGS2
SCHEMBL8774698 0.85 GAA (0.33) GAAMAPTPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-B1 PYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 1995-03-08 EP disclosed
WO-1991004248-A1 PYRIDINE DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-04-04 WO disclosed