SCHEMBL9159563

SCHEMBL9159563

N#Cc1ccc(C(c2ccc(C(F)(F)F)cc2)c2nc[nH]n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.47
CYP19A1 P11511 8/20 0.46
TRPM8 Q7Z2W7 1/20 0.39
CYP3A4 P08684 2/20 0.39
CYP3A5 P20815 2/20 0.39
VNN1 O95497 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
DGAT1 O75907 1/20 0.36
SOAT1 P35610 1/20 0.36
KCNH2 Q12809 1/20 0.36
MAOB P27338 2/20 0.36
KDM1A O60341 1/20 0.36
PRLHR P49683 2/20 0.34
DHODH Q02127 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1507799 0.89 CYP19A1 (0.46) CYP19A1CYP3A4
SCHEMBL9165274 0.82 ALDH1A1 (0.47) CYP19A1CYP3A4MAOBKDM1ADHODH
SCHEMBL8767389 0.82 CYP19A1 (0.41) CYP19A1CYP3A4MAOBKDM1A
SCHEMBL9165088 0.82 CA12 (0.47) CYP19A1
SCHEMBL9167057 0.80 CYP19A1 (0.47) CYP19A1VNN1MAOBKDM1A
SCHEMBL9158480 0.77 CYP19A1 (0.37) CYP19A1KDM1A
SCHEMBL9163386 0.76 AHR (0.38) CYP19A1TRPM8
SCHEMBL9163503 0.76 CYP19A1 (0.68) CYP19A1CYP3A4CYP3A5
SCHEMBL6474489 0.75 CYP19A1 (0.44) KIF11CYP19A1TRPM8CYP3A4CYP3A5
SCHEMBL1552746 0.75 CYP19A1 (0.38) CYP19A1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5473078-A Aromatase inhibiting compounds CIBA-GEIGY CORPORATION (US) 1995-12-05 US disclosed
US-5352795-A Condensing triazolylmethylbenzonitrile with fluorobenzonitrile under basic conditions using alkali metal alkoxide CIBA-GEIGY CORPORATION (US) 1994-10-04 US disclosed
US-5112845-A Inhibitors of estrogen synthesis, veterinary medicine CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
US-4978672-A Alpha-heterocyclc substituted tolunitriles CIBA-GEIGY CORPORATION (US) 1990-12-18 US disclosed