SCHEMBL8767389

SCHEMBL8767389

N#Cc1ccc(C(c2ccc(Br)cc2)c2nc[nH]n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 12/20 0.41
MAOB P27338 2/20 0.40
MAOA P21397 1/20 0.40
KDM1A O60341 2/20 0.34
IDO1 P14902 1/20 0.33
ERBB2 P04626 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP11B1 P15538 1/20 0.31
TSHR P16473 1/20 0.31
CYP11B2 P19099 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1507799 0.92 CYP19A1 (0.46) CYP19A1ALDH1A1CYP3A4CYP11B1TSHR
SCHEMBL9165274 0.85 ALDH1A1 (0.47) CYP19A1MAOBKDM1AERBB2ALDH1A1
SCHEMBL9165088 0.85 CA12 (0.47) CYP19A1
SCHEMBL9167057 0.83 CYP19A1 (0.47) CYP19A1MAOBMAOAKDM1AALDH1A1
SCHEMBL9159563 0.82 KIF11 (0.47) CYP19A1MAOBKDM1ACYP3A4
SCHEMBL9158480 0.81 CYP19A1 (0.37) CYP19A1KDM1AALDH1A1
SCHEMBL9165314 0.80 KDM4E (0.39) KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL9163503 0.80 CYP19A1 (0.68) CYP19A1KDM4EALDH1A1HPGDCYP3A4
SCHEMBL1552746 0.78 CYP19A1 (0.38) CYP19A1MAOBTSHR
SCHEMBL9160207 0.77 CYP19A1 (0.37) CYP19A1KDM1AALDH1A1CYP3A4CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0490816-B1 Fluoro-compounds and their use as aromatase inhibitors CIBA GEIGY AG (CH) 1997-07-09 EP disclosed
US-5637605-A ANTITUMOR AGENTS CIBA GEIGY CORPORATION (US) 1997-06-10 US disclosed
US-5583128-A ADMINISTERING A SIDE EFFECT REDUCED AROMATASE INHIBITOR CIBA-GEIGY CORPORATION (US) 1996-12-10 US disclosed
US-5473078-A Aromatase inhibiting compounds CIBA-GEIGY CORPORATION (US) 1995-12-05 US disclosed
US-5457209-A Antitumor agents CIBA-GEIGY CORPORATION (US) 1995-10-10 US disclosed
US-5376669-A Antitumor agents CIBA-GEIGY CORP. (US) 1994-12-27 US disclosed
US-5352795-A Condensing triazolylmethylbenzonitrile with fluorobenzonitrile under basic conditions using alkali metal alkoxide CIBA-GEIGY CORPORATION (US) 1994-10-04 US disclosed
US-5227393-A estrogen-dependent diseases, anticancer CIBA-GEIGY CORPORATION (US) 1993-07-13 US disclosed
EP-0490816-A2 Fluoro-compounds CIBA-GEIGY AG (CH) 1992-06-17 EP disclosed
US-5112845-A Inhibitors of estrogen synthesis, veterinary medicine CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
US-4978672-A Alpha-heterocyclc substituted tolunitriles CIBA-GEIGY CORPORATION (US) 1990-12-18 US disclosed