SCHEMBL9160695

SCHEMBL9160695

CCNC(=O)c1ccc2c(c1)NC=CC=C2

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 7/20 0.39
ALDH1A1 P00352 2/20 0.39
PDK2 Q15119 2/20 0.38
ALOX15 P16050 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CYP17A1 P05093 1/20 0.37
CYP3A4 P08684 1/20 0.37
RIPK1 Q13546 1/20 0.37
MAPK14 Q16539 1/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
RECQL P46063 1/20 0.36
CDK8 P49336 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5909057 0.71 CA12 (0.58) ALDH1A1NPC1RAB9ACA12CA9
SCHEMBL14157778 0.70 HPGDS (0.55) ALDH1A1NPC1RAB9ACYP17A1CYP3A4
SCHEMBL9713054 0.68 SMN1; SMN2 (0.67) ALDH1A1CYP1A2CYP2C19CDK8
SCHEMBL18083916 0.67 HDAC6 (0.60) ALDH1A1CA12CA9RECQLKDM4E
SCHEMBL4151138 0.67 NR1H4 (0.61) NPC1RAB9AMAPK14HPGD
SCHEMBL9979308 0.67 SMN1; SMN2 (0.48) ALDH1A1RAB9ACA12CA9HPGD
SCHEMBL1007936 0.67 LCK (0.37) ALDH1A1CYP3A4CYP2C19RECQLKDM4E
SCHEMBL4671199 0.67 CA1 (0.49) ALDH1A1ALOX15CA12CA9HPGD
SCHEMBL10851248 0.67 ALOX5 (0.48) ALDH1A1PDK2ALOX15NPC1RAB9A
SCHEMBL29528307 0.67 SMYD3 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0380355-B1 Carbamates of 6-chloro-7,8-dihydroxy-1-(4'-Hydroxyphenyl)-2,3,4,5-tetra-hydro-1H-3-benzazepine as prodrugs SMITHKLINE BEECHAM CORP (US) 1995-01-11 EP disclosed
EP-0380355-A2 Carbamates of 6-chloro-7,8-dihydroxy-1-(4'-Hydroxyphenyl)-2,3,4,5-tetra-hydro-1H-3-benzazepine as prodrugs SMITHKLINE BEECHAM CORPORATION (US) 1990-08-01 EP disclosed
US-4861771-A Carbamates of 6-chloro-7,8-dihydroxy-1-(4'-hydroxyphenyl)-2,3,4,5-tetrahydro-1H-3-benzazepine as prodrugs SMITHKLINE BECKMAN CORPORATION (US) 1989-08-29 US disclosed