SCHEMBL9165041

SCHEMBL9165041

N#Cc1ccc(C(c2nc[nH]n2)c2ccccc2O)cc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.37
TOP2B Q02880 1/20 0.37
CYP19A1 P11511 8/20 0.37
CYP11B1 P15538 2/20 0.34
OPRD1 P41143 1/20 0.32
GUSB P08236 1/20 0.32
CA12 O43570 1/20 0.31
CA2 P00918 1/20 0.31
CA3 P07451 1/20 0.31
CA6 P23280 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
MGAM O43451 1/20 0.31
GAA P10253 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1552746 0.86 CYP19A1 (0.38) TOP2ATOP2BCYP19A1OPRD1MGAM
SCHEMBL1507799 0.83 CYP19A1 (0.46) CYP19A1CYP11B1OPRD1CA12CA2
SCHEMBL9165088 0.82 CA12 (0.47) CYP19A1CA12CA2CA3CA6
SCHEMBL8767389 0.77 CYP19A1 (0.41) CYP19A1CYP11B1MAOB
SCHEMBL9165274 0.77 ALDH1A1 (0.47) CYP19A1MAOB
SCHEMBL9167057 0.75 CYP19A1 (0.47) CYP19A1GAAMAOB
SCHEMBL9163503 0.74 CYP19A1 (0.68) CYP19A1CYP11B1
SCHEMBL8110564 0.74 S1PR1 (0.34) CYP19A1GAA
SCHEMBL9163386 0.74 AHR (0.38) CYP19A1
SCHEMBL9165314 0.74 KDM4E (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5473078-A Aromatase inhibiting compounds CIBA-GEIGY CORPORATION (US) 1995-12-05 US disclosed
US-5352795-A Condensing triazolylmethylbenzonitrile with fluorobenzonitrile under basic conditions using alkali metal alkoxide CIBA-GEIGY CORPORATION (US) 1994-10-04 US disclosed
US-5112845-A Inhibitors of estrogen synthesis, veterinary medicine CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
US-4978672-A Alpha-heterocyclc substituted tolunitriles CIBA-GEIGY CORPORATION (US) 1990-12-18 US disclosed