SCHEMBL9166129

SCHEMBL9166129

C=CCCOc1ccc(C(=O)Oc2ccc(C#N)c(F)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 3/20 0.38
KMT2A Q03164 5/20 0.38
MEN1 O00255 2/20 0.38
LSS P48449 2/20 0.36
PRSS1 P07477 2/20 0.35
ACR P10323 2/20 0.35
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
KCNE1 P15382 1/20 0.35
KCNQ1 P51787 1/20 0.35
PLA2G7 Q13093 1/20 0.35
TRPV4 Q9HBA0 2/20 0.35
HTT P42858 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10429638 0.94 ALDH1A1 (0.51) ALDH1A1L3MBTL1MAPTKMT2AMEN1
SCHEMBL9164842 0.86 FFAR1 (0.35) ALDH1A1L3MBTL1KMT2AMEN1PRSS1
SCHEMBL9253512 0.86 ALDH1A1 (0.49) ALDH1A1L3MBTL1MAPTKMT2AMEN1
SCHEMBL10483910 0.85 MAPT (0.52) ALDH1A1MAPTKMT2APRSS1ACR
SCHEMBL10484072 0.85 MAPT (0.46) ALDH1A1L3MBTL1MAPTKMT2APRSS1
SCHEMBL9482558 0.84 ALDH1A1 (0.36) ALDH1A1L3MBTL1KMT2APRSS1ACR
SCHEMBL12604089 0.84 KMT2A (0.41) ALDH1A1MAPTKMT2AMEN1LSS
SCHEMBL7739126 0.84 CYP3A4 (0.41) ALDH1A1L3MBTL1MAPTKMT2AMEN1
SCHEMBL9166226 0.84 KDM1A (0.37) ALDH1A1
SCHEMBL10484028 0.83 LMNA (0.54) ALDH1A1MAPTKMT2APRSS1ACR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0464648-B1 4-Cyano-3-fluorophenyl esters HOFFMANN LA ROCHE (CH) 1995-12-06 EP disclosed
US-5413734-A 4-cyano-3-fluorophenyl esters HOFFMANN-LA ROCHE INC. (US) 1995-05-09 US disclosed
US-5185098-A Liquid crystalline mixtures containing 3,4-difluorophenyl-substituted bicyclohexyls HOFFMANN-LA ROCHE INC. (US) 1993-02-09 US disclosed
EP-0464648-A1 4-Cyano-3-fluorophenyl esters F. HOFFMANN-LA ROCHE AG (CH) 1992-01-08 EP disclosed