SCHEMBL9166226

SCHEMBL9166226

C=CCCc1ccc(-c2ccc(C(=O)Oc3ccc(C#N)c(F)c3)cc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 13/20 0.37
CYP11B2 P19099 3/20 0.35
CYP11B1 P15538 2/20 0.35
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
FFAR1 O14842 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
XDH P47989 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9164842 0.97 FFAR1 (0.35) KDM1ACYP11B2FFAR1FFAR4KDM4E
SCHEMBL9482558 0.90 ALDH1A1 (0.36) KDM1AFFAR1FFAR4ALDH1A1
SCHEMBL9162179 0.89 XDH (0.39) CYP11B2CYP11B1XDH
SCHEMBL7739126 0.85 CYP3A4 (0.41) ALDH1A1
SCHEMBL6567165 0.85 DAO (0.38) FFAR1FFAR4
SCHEMBL8048275 0.84 FFAR1 (0.36) KDM1ACYP11B2CYP11B1FFAR1FFAR4
SCHEMBL9166129 0.84 ALDH1A1 (0.43) ALDH1A1
SCHEMBL6567305 0.84 DAO (0.34) CYP11B2CYP11B1FFAR1FFAR4
SCHEMBL13198968 0.83 KMT2A (0.34) FFAR1FFAR4ALDH1A1HPGD
SCHEMBL16848606 0.83 CYP4A11 (0.39) KDM1AFFAR1FFAR4ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5413734-A 4-cyano-3-fluorophenyl esters HOFFMANN-LA ROCHE INC. (US) 1995-05-09 US disclosed