SCHEMBL9166552

SCHEMBL9166552

COc1ccc(-c2cnc3c(-c4cc(-c5ccccc5)cs4)cnn3c2O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.48
KMT2A Q03164 5/20 0.46
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
MAPT P10636 4/20 0.46
MEN1 O00255 3/20 0.46
STAT1 P42224 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
HPGD P15428 2/20 0.44
ALDH1A1 P00352 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FLT1 P17948 2/20 0.40
FLT4 P35916 2/20 0.40
BMP4 P12644 1/20 0.40
BACE1 P56817 1/20 0.40
LMNA P02545 2/20 0.39
RXFP1 Q9HBX9 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9170467 0.91 KDR (0.46) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9169606 0.90 RAB9A (0.47) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9166749 0.89 RAB9A (0.41) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9165874 0.88 HSD17B1 (0.44) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9173628 0.87 RAB9A (0.45) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9688673 0.86 NPC1 (0.47) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9171209 0.86 FYN (0.39) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9174113 0.85 CYP11B1 (0.41) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9165447 0.85 FYN (0.41) KDRKMT2ANPC1RAB9AMAPT
SCHEMBL9163418 0.85 GAK (0.39) KDRKMT2ANPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed