SCHEMBL9166576

SCHEMBL9166576

CCCOc1cccc(CC[S])c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
DHFR P00374 1/20 0.48
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CYP2D6 P10635 6/20 0.46
PPARG P37231 2/20 0.46
PPARA Q07869 2/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KCNH2 Q12809 2/20 0.44
GGPS1 O95749 1/20 0.43
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10235885 0.84 KMT2A (0.54) KMT2ADHFRCA1CA2CA7
SCHEMBL1047449 0.83 TAAR1 (0.64) KMT2ADHFRCA1CA2CA7
SCHEMBL18427030 0.83 LMNA (0.53) KMT2ADHFRCYP2D6SMN1; SMN2KCNH2
SCHEMBL8046926 0.83 KMT2A (0.57) KMT2ADHFRCA1CA2CA7
SCHEMBL9166584 0.83 DHFR (0.51) KMT2ADHFRCA1CA2CA7
SCHEMBL3811700 0.83 CYP4F2 (0.63) KMT2ADHFRCA1CA2CA7
SCHEMBL7853630 0.83 KMT2A (0.49) KMT2ADHFRCA1CA2CA7
SCHEMBL59488 0.82 KDM4E (0.61) KMT2ADHFRKDM4EALDH1A1SMN1; SMN2
SCHEMBL10236068 0.81 PPARA (0.67) CYP2D6PPARGPPARAKCNH2GGPS1
SCHEMBL8957636 0.81 PPARA (0.67) CYP2D6PPARGPPARAKCNH2GGPS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed