SCHEMBL9167579

SCHEMBL9167579

CCOC([C]=O)c1ccccc1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.42
CYP2D6 P10635 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
SLC22A2 O15244 1/20 0.36
SLC22A1 O15245 1/20 0.36
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
ADRA2A P08913 1/20 0.36
CHRM1 P11229 1/20 0.36
ADRA2B P18089 1/20 0.36
CHRM3 P20309 1/20 0.36
DRD1 P21728 1/20 0.36
HRH2 P25021 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9167590 1.00 ESR1 (0.42) ESR1CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL9167586 1.00 ESR1 (0.42) ESR1CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL9160666 0.81 CYP3A4 (0.38) SLC6A2SLC6A4CYP3A4CYP2C9L3MBTL1
SCHEMBL9160673 0.81 CYP3A4 (0.38) SLC6A2SLC6A4CYP3A4CYP2C9L3MBTL1
SCHEMBL9160678 0.81 CYP3A4 (0.38) SLC6A2SLC6A4CYP3A4CYP2C9L3MBTL1
SCHEMBL9160194 0.79 ESR1 (0.47) ESR1CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL9160198 0.79 ESR1 (0.47) ESR1CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL9160191 0.79 ESR1 (0.47) ESR1CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL9165582 0.76 L3MBTL1 (0.43) CYP2D6SLC6A2SLC6A4SLC6A3CHRM2
SCHEMBL8536881 0.76 L3MBTL1 (0.43) CYP2D6SLC6A2SLC6A4SLC6A3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469887-B1 Acetamide derivatives ZENECA LTD (GB) 1994-12-14 EP claimed
US-5270342-A Acetamide derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US claimed
US-5430060-A Aldose reductase inhibitor ZENECA LIMITED (GB) 1995-07-04 US disclosed
US-5270342-A Acetamide derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed