SCHEMBL9167775

SCHEMBL9167775

CSC(=O)c1ccc(-c2ccccc2)c(O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.53
CNR2 P34972 3/20 0.51
ALOX5 P09917 1/20 0.48
BACE1 P56817 1/20 0.45
ESR2 Q92731 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
BCL2L1 Q07817 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PTGS2 P35354 2/20 0.40
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B1 P14061 1/20 0.39
CNR1 P21554 1/20 0.39
HPGDS O60760 1/20 0.38
PTPN1 P18031 1/20 0.38
ABCC1 P33527 1/20 0.38
KDM4E B2RXH2 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9166730 0.85 ESR2 (0.56) EGFRCNR2ESR2ALDH1A1PTGS2
SCHEMBL9163491 0.81 MKNK1 (0.50) EGFRALDH1A1PTGS2ABCC1CA12
SCHEMBL9436727 0.81 PTGS2 (0.46) EGFRPTGS2
SCHEMBL3663963 0.80 POLB (0.59) EGFRCNR2ALOX5BACE1ALDH1A1
SCHEMBL9170977 0.77 SMN1; SMN2 (0.59) ALDH1A1HPGDMAPTSMN1; SMN2PTPN1
SCHEMBL14832783 0.76 EGFR (0.79) EGFRCNR2ALOX5ALDH1A1HPGD
SCHEMBL812709 0.72 KMT2A (0.56) ALDH1A1HPGDHSD17B10MAPTSMN1; SMN2
SCHEMBL9488109 0.72 CA12 (0.66) EGFRCNR2ESR2ALDH1A1MAPT
SCHEMBL29914657 0.72 EGFR (0.56) EGFRCNR2ALOX5BACE1ESR2
SCHEMBL11665321 0.72 EGFR (0.56) EGFRALDH1A1PTGS2SMN1; SMN2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269859-B2 Pyrazolotriazine compounds OTSUKA PHARMA CO LTD (JP) 1995-10-18 EP disclosed
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed
US-4824834-A TREATING GOUT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-04-25 US disclosed
EP-0269859-A2 Pyrazolotriazine compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-06-08 EP disclosed