SCHEMBL9436727

SCHEMBL9436727

CSC(=O)c1ccc(-c2ccccc2)c(S(C)(=O)=O)c1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.46
ROCK2 O75116 1/20 0.44
LOXL2 Q9Y4K0 2/20 0.42
PTGDR2 Q9Y5Y4 2/20 0.40
TDP1 Q9NUW8 1/20 0.39
EGFR P00533 1/20 0.38
BCAT2 O15382 1/20 0.38
ACLY P53396 1/20 0.37
GSTO1 P78417 1/20 0.37
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8796477 0.86 TDP1 (0.50) PTGS2ROCK2LOXL2TDP1ACLY
SCHEMBL16618470 0.83 PTGS2 (0.47) PTGS2ROCK2LOXL2BCAT2ACLY
SCHEMBL9167775 0.81 EGFR (0.53) PTGS2EGFR
SCHEMBL9166730 0.80 ESR2 (0.56) PTGS2ROCK2EGFR
SCHEMBL9436730 0.77 PTGS2 (0.50) PTGS2ROCK2LOXL2PTGDR2TDP1
Hydrochloric Acid SCHEMBL8895292 0.76 SLC9A1 (0.59)
SCHEMBL9163491 0.76 MKNK1 (0.50) PTGS2ROCK2EGFR
SCHEMBL27765267 0.76 ALOX5 (0.55) PTGS2LOXL2PTGDR2ACLY
SCHEMBL9189128 0.74 SLC9A1 (0.46) LOXL2
Hydrochloric Acid SCHEMBL8895287 0.74 ROCK2 (0.46) PTGS2ROCK2LOXL2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292755-A USPA benzolyguanidines HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-08 US disclosed
US-5091394-A BENZOYLGUANIDINES, A PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-25 US disclosed