SCHEMBL9166730

SCHEMBL9166730

CSC(=O)c1ccc(-c2ccccc2)c(C)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.56
HSD17B1 P14061 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
RARB P10826 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
OXTR P30559 2/20 0.42
AVPR1A P37288 2/20 0.42
AVPR2 P30518 1/20 0.42
AVPR1B P47901 1/20 0.42
EGFR P00533 1/20 0.41
ADH5 P11766 1/20 0.41
SLC2A1 P11166 1/20 0.41
LDHA P00338 1/20 0.41
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
EPHX1 P07099 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9167775 0.85 EGFR (0.53) ESR2HSD17B1L3MBTL1EGFRCNR2
SCHEMBL29707122 0.82 ESR2 (0.58) ESR2HSD17B1L3MBTL1RARBADH5
SCHEMBL121338 0.82 ESR2 (0.58) ESR2HSD17B1L3MBTL1RARBADH5
Hydrochloric Acid SCHEMBL5753140 0.81 ESR2 (0.56) ESR2HSD17B1L3MBTL1RARBADH5
SCHEMBL5608472 0.81 HSD17B1 (0.62) ESR2HSD17B1L3MBTL1PPARGPPARA
SCHEMBL9163491 0.80 MKNK1 (0.50) AVPR1AAVPR2EGFRPTGS2ALDH1A1
SCHEMBL9436727 0.80 PTGS2 (0.46) EGFRPTGS2ROCK2
SCHEMBL8906586 0.79 ESR2 (0.55) ESR2HSD17B1L3MBTL1PPARGPPARA
SCHEMBL9164912 0.79 ESR2 (0.55) ESR2HSD17B1L3MBTL1PPARGPPARA
SCHEMBL537623 0.79 CNR2 (0.60) ESR2HSD17B1L3MBTL1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269859-B2 Pyrazolotriazine compounds OTSUKA PHARMA CO LTD (JP) 1995-10-18 EP disclosed
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed
US-4824834-A TREATING GOUT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-04-25 US disclosed
EP-0269859-A2 Pyrazolotriazine compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-06-08 EP disclosed