SCHEMBL9168977

SCHEMBL9168977

O=C(C#CI)Nc1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.52
HTT P42858 5/20 0.51
MAPT P10636 3/20 0.51
TSHR P16473 2/20 0.51
LMNA P02545 2/20 0.51
NLRP3 Q96P20 2/20 0.51
ALDH1A1 P00352 3/20 0.48
KMT2A Q03164 6/20 0.46
MEN1 O00255 5/20 0.46
RAB9A P51151 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 2/20 0.44
EPHX1 P07099 2/20 0.44
CHRM1 P11229 2/20 0.44
NLRP1 Q9C000 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
SLC6A2 P23975 1/20 0.44
PDE4A P27815 1/20 0.44
EPHX2 P34913 1/20 0.44
ADRA1A P35348 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950876 0.82 NPC1 (0.53) NPC1HTTMAPTTSHRLMNA
SCHEMBL8950841 0.81 NPC1 (0.52) NPC1HTTMAPTTSHRLMNA
SCHEMBL9164150 0.80 EPHX2 (0.52) NPC1MAPTTSHRNLRP3KMT2A
SCHEMBL8950777 0.76 NPC1 (0.55) NPC1HTTMAPTTSHRLMNA
SCHEMBL9169249 0.75 USP2 (0.50) NPC1MAPTALDH1A1KMT2ARAB9A
SCHEMBL15443343 0.73 ALDH1A1 (0.45) NPC1HTTMAPTTSHRLMNA
SCHEMBL15691175 0.73 NPC1 (0.61) NPC1HTTMAPTTSHRLMNA
SCHEMBL11048619 0.72 MEN1 (0.76) NPC1HTTMAPTTSHRLMNA
SCHEMBL21568080 0.72 NPC1 (0.67) NPC1HTTMAPTTSHRLMNA
SCHEMBL4741253 0.72 MEN1 (0.76) NPC1HTTMAPTTSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519427-B1 N-substituted-3-iodopropiolamide, production and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-04-26 EP disclosed
EP-0552418-A1 N-substituted-3-iodopropiolamide, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-07-28 EP disclosed
EP-0519427-A2 N-substituted-3-iodopropiolamide, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-23 EP disclosed