SCHEMBL8950841

SCHEMBL8950841

O=C(C#CBr)Nc1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.52
ALDH1A1 P00352 3/20 0.48
HTT P42858 6/20 0.47
LMNA P02545 3/20 0.47
MAPT P10636 3/20 0.47
TSHR P16473 2/20 0.47
NLRP3 Q96P20 2/20 0.47
POLB P06746 1/20 0.46
KMT2A Q03164 6/20 0.46
MEN1 O00255 5/20 0.46
RAB9A P51151 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
EPHX1 P07099 2/20 0.44
CHRM1 P11229 2/20 0.44
NLRP1 Q9C000 1/20 0.44
GAA P10253 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
SLC6A2 P23975 1/20 0.44
PDE4A P27815 1/20 0.44
EPHX2 P34913 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950876 0.82 NPC1 (0.53) NPC1ALDH1A1HTTLMNAMAPT
SCHEMBL9168977 0.81 NPC1 (0.52) NPC1ALDH1A1HTTLMNAMAPT
SCHEMBL8950880 0.79 MEN1 (0.61) NPC1ALDH1A1HTTLMNAMAPT
SCHEMBL8950777 0.76 NPC1 (0.55) NPC1ALDH1A1HTTLMNAMAPT
SCHEMBL8950904 0.75 RAB9A (0.49) NPC1ALDH1A1RAB9AMAPK1
SCHEMBL15443343 0.73 ALDH1A1 (0.45) NPC1ALDH1A1HTTLMNAMAPT
SCHEMBL11048619 0.72 MEN1 (0.76) NPC1ALDH1A1HTTLMNAMAPT
SCHEMBL4741253 0.72 MEN1 (0.76) NPC1ALDH1A1HTTLMNAMAPT
SCHEMBL21568080 0.72 NPC1 (0.67) NPC1ALDH1A1HTTLMNAMAPT
SCHEMBL3912100 0.70 NPC1 (0.64) NPC1ALDH1A1HTTLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5538998-A PEST CONTROL AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US claimed
EP-0649835-A1 Halopropiolamide compound, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-04-26 EP claimed
US-5538998-A PEST CONTROL AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
EP-0649835-A1 Halopropiolamide compound, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-04-26 EP disclosed