SCHEMBL9169871

SCHEMBL9169871

COC(=S)c1cc(C)cc(O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.50
ALDH1A1 P00352 1/20 0.48
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
PTPN1 P18031 1/20 0.35
CNR2 P34972 1/20 0.33
CYP3A4 P08684 3/20 0.32
ACHE P22303 2/20 0.32
ATM Q13315 1/20 0.32
TPMT P51580 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CA5A P35218 1/20 0.32
MAPT P10636 1/20 0.31
RET P07949 1/20 0.31
KIF5B P33176 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5380375 0.87 TPMT (0.42) ALDH1A1CNR2ATMTPMTTDP1
SCHEMBL13892529 0.75 HCAR1 (0.50) HCAR1ALDH1A1CA12CA1CA2
SCHEMBL31208002 0.75 CA12 (0.76) HCAR1ALDH1A1CA12CA1CA2
SCHEMBL2259905 0.75 CA12 (0.76) HCAR1ALDH1A1CA12CA1CA2
Orcinol SCHEMBL998779 0.71 ALDH1A1 (0.71) HCAR1ALDH1A1CA12CA1CA2
SCHEMBL27481953 0.71 HDAC8 (0.50) ALDH1A1ACHEMAPT
SCHEMBL8920001 0.69 HCAR1 (0.48) HCAR1ALDH1A1ACHEATMTDP1
SCHEMBL31211908 0.69 ATM (0.61) ALDH1A1ATMTDP1
SCHEMBL10370027 0.69 HCAR1 (0.71) HCAR1ALDH1A1CA12CA1CA2
SCHEMBL9436697 0.69 TDP1 (0.54) ALDH1A1ACHETDP1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5446189-A Diester intermediates for diacid enzyme inhibitor HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed
US-5324747-A Treatment of inflammatory diseases HOFFMANN-LA ROCHE INC. (US) 1994-06-28 US disclosed
EP-0579066-A2 N-substituted anilines F. HOFFMANN-LA ROCHE AG (CH) 1994-01-19 EP disclosed