SCHEMBL9169977

SCHEMBL9169977

COc1ccc(CCC(C)NC(=O)Cc2ccc(OC)c(OC)c2)cc1

nearest known ligand 0.79

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.79
MEN1 O00255 5/20 0.79
ALDH1A1 P00352 5/20 0.71
MAPT P10636 2/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
HTT P42858 3/20 0.56
LMNA P02545 2/20 0.56
NPC1 O15118 1/20 0.56
GAA P10253 2/20 0.52
TAS1R3 Q7RTX0 1/20 0.52
TAS1R1 Q7RTX1 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
POLB P06746 1/20 0.51
MAPK1 P28482 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14399043 0.91 ALDH1A1 (0.73) KMT2AMEN1ALDH1A1TAS1R3TAS1R1
SCHEMBL5323935 0.84 ALDH1A1 (0.66) KMT2AMEN1ALDH1A1TAS1R3TAS1R1
SCHEMBL9829926 0.83 KMT2A (0.65) KMT2AMEN1MAPTCYP3A4CYP2D6
SCHEMBL9829918 0.83 KMT2A (0.65) KMT2AMEN1MAPTCYP3A4CYP2D6
SCHEMBL11808978 0.81 KMT2A (0.65) KMT2AMEN1ALDH1A1MAPTHTT
SCHEMBL8259636 0.81 KMT2A (0.62) KMT2AMEN1ALDH1A1MAPTCYP3A4
SCHEMBL25306507 0.78 ALDH1A1 (0.72) KMT2AMEN1ALDH1A1MAPTHTT
SCHEMBL9164083 0.78 HTT (0.78) KMT2AMEN1MAPTCYP3A4CYP2D6
SCHEMBL9164074 0.78 HTT (0.78) KMT2AMEN1MAPTCYP3A4CYP2D6
SCHEMBL19427446 0.78 EPHX2 (0.80) KMT2AMEN1ALDH1A1MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0443606-B1 4-(4-alkoxyphenyl)-2-butylamine derivatives and process therefor SHIONOGI & CO (JP) 1995-05-10 EP disclosed
US-5073648-A Intermediates for dopamine derivatives SHIONOGI & CO., LTD. (JP) 1991-12-17 US disclosed
EP-0443606-A2 4-(4-alkoxyphenyl)-2-butylamine derivatives and process therefor SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1991-08-28 EP disclosed
US-3987200-A INOTROPIC AGENTS, 3,4-DIHYDROXY-PHENYL-ALKYL PHENETHYLAMINE ELI LILLY AND COMPANY (US) 1976-10-19 US disclosed