SCHEMBL9170664

SCHEMBL9170664

COCCOCOCc1cccc2c1Cc1c(C(=O)O)nn(-c3ccccc3)c1-2

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 13/20 0.39
PIK3R2 O00459 13/20 0.39
PIK3CA P42336 13/20 0.39
PIK3CB P42338 13/20 0.39
PIK3CG P48736 13/20 0.39
PIK3R5 Q8WYR1 13/20 0.39
PIK3R3 Q92569 13/20 0.39
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CCNA1 P78396 1/20 0.38
F10 P00742 1/20 0.37
CACNA1G O43497 2/20 0.35
CACNA1H O95180 2/20 0.35
RIPK1 Q13546 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9256845 0.93 PIK3CD (0.38) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9173465 0.90 ALDH1A1 (0.45) CCNA2CDK2CCNA1F10
SCHEMBL9837911 0.82 PIK3CD (0.33) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9522531 0.75 MAPT (0.43)
SCHEMBL9173375 0.72 ALDH1A1 (0.51) CCNA2CDK2CCNA1F10
SCHEMBL9172754 0.70 PTGER1 (0.47) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9170672 0.70 PIK3CD (0.42) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9170065 0.69 ALDH1A1 (0.52) CCNA2CDK2CCNA1
SCHEMBL9523022 0.69 MAPT (0.42)
SCHEMBL30433314 0.68 TSHR (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5424308-A Immunomodulating agents FARMITALIA CARLO ERBA S.R.L. (IT) 1995-06-13 US disclosed
EP-0422051-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-04-17 EP disclosed
WO-1989012630-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed
EP-0347773-A1 Condensed Pyrazole 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1989-12-27 EP disclosed