SCHEMBL9256845

SCHEMBL9256845

COCCOCOCc1cccc2c1Cc1c(C(=O)Cl)nn(-c3ccccc3)c1-2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 13/20 0.38
PIK3R2 O00459 13/20 0.38
PIK3CA P42336 13/20 0.38
PIK3CB P42338 13/20 0.38
PIK3CG P48736 13/20 0.38
PIK3R5 Q8WYR1 13/20 0.38
PIK3R3 Q92569 13/20 0.38
RIPK1 Q13546 1/20 0.35
CACNA1G O43497 2/20 0.34
CACNA1H O95180 2/20 0.34
GRM5 P41594 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
F10 P00742 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9170664 0.93 PIK3CD (0.39) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9173465 0.88 ALDH1A1 (0.45) ALDH1A1CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL9837911 0.81 PIK3CD (0.33) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9523022 0.76 MAPT (0.42) MAPT
SCHEMBL9166215 0.72 CCNA2 (0.44) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9173375 0.71 ALDH1A1 (0.51) ALDH1A1CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL9174527 0.70 ALDH1A1 (0.50) ALDH1A1CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL9522531 0.69 MAPT (0.43) MAPT
SCHEMBL8588667 0.67 CCNA2 (0.49) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9736649 0.66 TP53 (0.42) ALDH1A1CYP3A4MAPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5424308-A Immunomodulating agents FARMITALIA CARLO ERBA S.R.L. (IT) 1995-06-13 US disclosed
EP-0422051-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-04-17 EP disclosed
WO-1989012630-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed
EP-0347773-A1 Condensed Pyrazole 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1989-12-27 EP disclosed