SCHEMBL9172018

SCHEMBL9172018

COc1cccc(Cc2cnc3c(-c4cc(-c5ccccc5)cs4)cnn3c2O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.39
KDR P35968 2/20 0.38
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 2/20 0.37
CYP3A4 P08684 4/20 0.36
PRKACA P17612 3/20 0.36
ROCK1 Q13464 3/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
GAA P10253 1/20 0.36
LTA4H P09960 1/20 0.36
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9167960 0.93 KDR (0.36) KDRCYP11B1CYP11B2ALDH1A1MEN1
SCHEMBL9174113 0.91 CYP11B1 (0.41) KDRCYP11B1CYP11B2ALDH1A1MEN1
SCHEMBL9166631 0.89 NPC1 (0.36) CYP11B1CYP11B2ALDH1A1MEN1KMT2A
SCHEMBL9169535 0.88 HSD17B1 (0.39) DHFRKDRCYP3A4MEN1KMT2A
SCHEMBL9170467 0.85 KDR (0.46) KDRCYP3A4ALDH1A1MEN1KMT2A
SCHEMBL9170993 0.84 GAK (0.35) KDRLTA4HALDH1A1MEN1KMT2A
SCHEMBL9171199 0.84 HSD17B1 (0.38) KDRCYP3A4MEN1KMT2AMAPT
SCHEMBL9172217 0.82 NPC1 (0.36) KDRALDH1A1MEN1KMT2AMAPT
SCHEMBL9172004 0.82 DHFR (0.41) DHFRKDRCYP11B1CYP11B2GAA
SCHEMBL9170564 0.82 NPC1 (0.41) KDRALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed