SCHEMBL9170993

SCHEMBL9170993

COc1ccccc1Cc1cnc2c(-c3cc(-c4ccccc4)cs3)cnn2c1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 1/20 0.35
PTGER1 P34995 4/20 0.35
PTGER4 P35408 4/20 0.35
PTGER3 P43115 4/20 0.35
PTGER2 P43116 4/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 2/20 0.34
RELA Q04206 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
FYN P06241 2/20 0.34
LTA4H P09960 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
STAT1 P42224 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9170543 0.87 RAB9A (0.35) PTGER1PTGER4PTGER3PTGER2MAPT
SCHEMBL9163418 0.86 GAK (0.39) GAKMAPTNPC1RAB9ANFKB1
SCHEMBL9174113 0.86 CYP11B1 (0.41) MAPTNPC1RAB9ASMN1; SMN2FYN
SCHEMBL9167960 0.86 KDR (0.36) MAPTNPC1RAB9ANFKB1NFKB2
SCHEMBL9166631 0.85 NPC1 (0.36) PTGER1PTGER4PTGER3PTGER2MAPT
SCHEMBL9172018 0.84 DHFR (0.39) MAPTSMN1; SMN2FYNLTA4HKDM4E
SCHEMBL9171209 0.84 FYN (0.39) GAKMAPTNPC1RAB9AFYN
SCHEMBL9170564 0.84 NPC1 (0.41) PTGER1PTGER4PTGER3PTGER2MAPT
SCHEMBL9171199 0.82 HSD17B1 (0.38) PTGER1PTGER4PTGER3PTGER2MAPT
SCHEMBL9173574 0.81 RAB9A (0.39) PTGER1PTGER4PTGER3PTGER2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed