SCHEMBL9177629

SCHEMBL9177629

CCOC(=O)CN1C(=O)/C(=N/OC)c2cc(Br)ccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
CUL4A Q13619 1/20 0.48
UCHL1 P09936 2/20 0.48
UCHL3 P15374 2/20 0.48
PIN1 Q13526 1/20 0.46
PIN4 Q9Y237 1/20 0.46
RXFP1 Q9HBX9 1/20 0.45
CES1 P23141 1/20 0.44
MAPT P10636 3/20 0.44
HTT P42858 3/20 0.44
HSD17B10 Q99714 1/20 0.44
PPARG P37231 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRA6 Q16445 1/20 0.41
GSK3A P49840 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9177631 1.00 ALDH1A1 (0.54) ALDH1A1CUL4AUCHL1UCHL3PIN1
SCHEMBL6316299 0.88 ALDH1A1 (0.56) ALDH1A1CUL4AUCHL1UCHL3PIN1
SCHEMBL6316296 0.88 ALDH1A1 (0.56) ALDH1A1CUL4AUCHL1UCHL3PIN1
SCHEMBL12674685 0.83 ALDH1A1 (0.76) ALDH1A1CUL4APIN1PIN4RXFP1
SCHEMBL6319755 0.82 ALDH1A1 (0.46) ALDH1A1PIN1PIN4RXFP1MAPT
SCHEMBL6323847 0.82 ALDH1A1 (0.46) ALDH1A1PIN1PIN4RXFP1MAPT
SCHEMBL6316140 0.79 ALDH1A1 (0.55) ALDH1A1UCHL1UCHL3CES1MAPT
SCHEMBL6316144 0.79 ALDH1A1 (0.55) ALDH1A1UCHL1UCHL3CES1MAPT
SCHEMBL522944 0.76 PIN1 (0.68) ALDH1A1PIN1PIN4RXFP1MAPT
SCHEMBL30892347 0.74 UCHL1 (0.42) ALDH1A1CUL4AUCHL1UCHL3CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432648-B1 Isatine derivatives, their preparation and use NEUROSEARCH AS (DK) 1995-08-02 EP disclosed
US-5198461-A Isatine derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-30 US disclosed
EP-0432648-A2 Isatine derivatives, their preparation and use NEUROSEARCH A/S (DK) 1991-06-19 EP disclosed