SCHEMBL9185044

SCHEMBL9185044

COC(C)(C)Oc1ccccc1CC#N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.35
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
RIPK1 Q13546 2/20 0.33
NPC1 O15118 1/20 0.33
THRB P10828 1/20 0.33
RAB9A P51151 1/20 0.33
IDO1 P14902 2/20 0.33
TAAR1 Q96RJ0 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
SLC6A4 P31645 1/20 0.31
KMT2A Q03164 1/20 0.31
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA4 P22748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9182573 0.78 APLNR (0.41) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL198463 0.78 IDO1 (0.52) ALDH1A1TSHRGAAMAPTIDO1
SCHEMBL625370 0.77 GRIN2B (0.40) ALDH1A1HPGDGAASLC6A4
SCHEMBL29921250 0.77 GRIN2B (0.40) ALDH1A1HPGDGAASLC6A4
SCHEMBL6544128 0.76 ALDH1A1 (0.51) ALDH1A1HPGDTSHRMAPTKMT2A
SCHEMBL8095035 0.73 KCNH2 (0.37) ALDH1A1HPGDTSHRGAAMAPT
SCHEMBL8595493 0.72 HTT (0.47) ALDH1A1TSHRGAAMAPTNPC1
SCHEMBL7825335 0.72 ALDH1A1 (0.36) ALDH1A1HPGDTSHRRIPK1IDO1
SCHEMBL7197450 0.72 L3MBTL1 (0.55) ALDH1A1HPGDTSHRGAAMAPT
Ammonia Solution, Strong SCHEMBL3938120 0.71 IDO1 (0.44) ALDH1A1TSHRGAAMAPTIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5412119-A Method of preparing vicinal aminoalcohols DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1995-05-02 US disclosed
EP-0558824-A1 Method for the preparation of vicinal aminoalcohols and optically active O-protected derivatives thereof DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1993-09-08 EP disclosed
EP-0554933-A1 Method of preparing vicinal aminoalcohols DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1993-08-11 EP disclosed