SCHEMBL9190822

SCHEMBL9190822

CCc1cc(SC[Si](C)(C)CSc2cc(CC)c(O)c(CC)c2)cc(CC)c1O

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
DHFR P00374 2/20 0.34
SIRT1 Q96EB6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8575917 0.89 GABRA1 (0.39) GABRA1GABRB2CYP1A2CYP3A4CYP2C9
SCHEMBL9193207 0.85 DHFR (0.35) DHFR
SCHEMBL9195084 0.83 GABRA1 (0.38) GABRA1GABRB2CYP1A2CYP3A4CYP2C9
SCHEMBL9195092 0.82 TYR (0.39) GABRA1GABRB2CYP3A4
SCHEMBL9190294 0.81 GABRA1 (0.33) GABRA1GABRB2CYP1A2CYP3A4CYP2C9
SCHEMBL9191120 0.80 GABRA1 (0.44) GABRA1GABRB2
SCHEMBL8579964 0.80 GABRA1 (0.39) GABRA1GABRB2CYP1A2CYP3A4CYP2C9
SCHEMBL8578127 0.79 GABRA1 (0.39) GABRA1GABRB2SIRT1
SCHEMBL9193227 0.76 CA1 (0.41) CYP1A2CYP3A4CYP2C9
SCHEMBL2678101 0.74 GABRA1 (0.48) GABRA1GABRB2CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0464844-B1 Novel bis (4-(2,6-di-alkyl)phenol)silane derivatives as antiatherosclerotic agents and as antioxidants MERRELL DOW PHARMA (US) 1995-12-27 EP disclosed
US-5281738-A Anticholesterol agents MERRELL DOW PHARMACEUTICALS INC. (US) 1994-01-25 US disclosed
EP-0464844-A1 Novel bis (4-(2,6-di-alkyl)phenol)silane derivatives as antiatherosclerotic agents and as antioxidants MERRELL DOW PHARMACEUTICALS INC. (US) 1992-01-08 EP disclosed