SCHEMBL9192247

SCHEMBL9192247

CC1(C)CCSc2cc[c]cc21

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RARA P10276 8/20 0.37
RARB P10826 8/20 0.37
RARG P13631 8/20 0.37
RXRA P19793 2/20 0.37
CYP3A4 P08684 2/20 0.34
CYP26A1 O43174 1/20 0.34
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811695 0.78
SCHEMBL7804624 0.76
SCHEMBL7814778 0.73 ESR2 (0.30)
SCHEMBL1649848 0.73 RARA (0.40) RARARARBRARGRXRACYP3A4
SCHEMBL2014128 0.72 RXRA (0.33) RARARARBRARGRXRACYP3A4
SCHEMBL9843477 0.71 RARA (0.37) RARARARBRARG
SCHEMBL8560479 0.70 RARA (0.34) RARARARBRARGRXRACYP3A4
SCHEMBL8293245 0.69 RARA (0.47) RARARARBRARGRXRACYP3A4
SCHEMBL816209 0.68
SCHEMBL9054284 0.68 RARA (0.46) RARARARBRARGRXRACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0405028-B1 Thiochroman esters of phenols and terephthalates having retinoid-like activity ALLERGAN INC (US) 1995-10-11 EP claimed
EP-0405028-A1 Thiochroman esters of phenols and terephthalates having retinoid-like activity ALLERGAN, INC (US) 1991-01-02 EP claimed
US-4895868-A PSORIASIS, SKIN DISORDERS, ANTIARTHRITIC, WOUND HEALING, EYE DRYNESS ALLERGAN, INC. (US) 1990-01-23 US claimed
EP-0682516-A1 THERAPEUTIC USE OF COMPOUNDS HAVING SELECTIVE AGONIST-LIKE ACTIVITY ON RXR RETINOID RECEPTORS ALLERGAN, INC. (US) 1995-11-22 EP disclosed
WO-1994017796-A1 THERAPEUTIC USE OF COMPOUNDS HAVING SELECTIVE AGONIST-LIKE ACTIVITY ON RXR RETINOID RECEPTORS ALLERGAN, INC. (US) 1994-08-18 WO disclosed
US-5324840-A Skin disorders ALLERGAN, INC. (US) 1994-06-28 US disclosed
EP-0263492-B1 RETINOIDS, THEIR PREPARATION AND USE AS PHARMACEUTICAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-03-13 EP disclosed
US-4900478-A SKIN DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-02-13 US disclosed
EP-0263492-A1 Retinoids, their preparation and use as pharmaceutical compounds F. HOFFMANN-LA ROCHE AG (CH) 1988-04-13 EP disclosed