SCHEMBL8560479

SCHEMBL8560479

Cc1[c]cc2c(c1)SCCC2(C)C

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RARA P10276 8/20 0.34
RARB P10826 8/20 0.34
RARG P13631 8/20 0.34
RXRA P19793 2/20 0.34
CYP3A4 P08684 2/20 0.31
CYP26A1 O43174 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL330266 0.74 RXRA (0.35) RARARARBRARGRXRACYP26A1
SCHEMBL6668874 0.71 EPHX2 (0.39) RARARARBRARGRXRACYP3A4
SCHEMBL9192247 0.70 RARA (0.37) RARARARBRARGRXRACYP3A4
SCHEMBL9092256 0.69 RARA (0.36) RARARARBRARGRXRACYP3A4
SCHEMBL9054107 0.69 RARA (0.36) RARARARBRARGRXRACYP3A4
SCHEMBL6665606 0.69 RARA (0.36) RARARARBRARGRXRACYP3A4
SCHEMBL8293245 0.68 RARA (0.47) RARARARBRARGRXRACYP3A4
SCHEMBL10515346 0.67 RXRA (0.39) RXRA
SCHEMBL19259616 0.67 RARA (0.37) RARARARBRARGRXRACYP3A4
SCHEMBL9054573 0.67 RARA (0.37) RARARARBRARGRXRACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5717094-A 6-THIOCHROMANYL-ETHYNE, 6-CHROMANYL ETHYNE AND 6-TETRAHYDROQUINOLINYL ETHYNE OR THEIR METAL SALTS ARE REACTED WITH SUITABLE HALO SUBSTITUTED PHENYL OR HETEROARYL COMPUNDS ALLERGAN (US) 1998-02-10 US disclosed
US-5248777-A Inhibitors of ornithine decarboxylase ALLERGAN, INC. (US) 1993-09-28 US disclosed
US-5053523-A Chemical intermediate for compounds having retinoic acid-like activity ALLERGAN, INC. (US) 1991-10-01 US disclosed
US-5023341-A Acetylene thiochroman ALLERGAN, INC. (US) 1991-06-11 US disclosed