SCHEMBL9195166

SCHEMBL9195166

O=C1c2ccccc2C2(c3cccc4c3CCC4)OCCN12

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
PARP1 P09874 7/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CES1 P23141 2/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SIGMAR1 Q99720 2/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
AVPR1A P37288 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9196504 0.97 NPC1 (0.39) CYP2A6MAOAMAOBNPC1POLB
SCHEMBL9201268 0.95 CYP2A6 (0.38) CYP2A6MAOAMAOBNPC1POLB
SCHEMBL9225508 0.81 MAPT (0.39) CYP2A6MAOAMAOBPOLBPARP1
SCHEMBL9196127 0.79 NPC1 (0.51) NPC1POLBMEN1KMT2AHTT
SCHEMBL9197570 0.79 PARP1 (0.43) NPC1POLBPARP1KMT2AHTT
SCHEMBL9199522 0.77 SLC6A3 (0.40) NPC1POLBMEN1KMT2AHTT
SCHEMBL9199731 0.76 NPC1 (0.40) NPC1POLBPARP1MEN1KMT2A
SCHEMBL9200340 0.75 NPC1 (0.36) NPC1POLBPARP1MEN1KMT2A
SCHEMBL9205975 0.75 CYP2A6 (0.38) CYP2A6MAOAMAOBNPC1POLB
SCHEMBL9280066 0.75 CHRM5 (0.46) NPC1POLBHTTSMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0575425-B1 USE OF OXAZOLO- 2,3-a]ISOINDOLE AND IMIDAZO 2,1-a]ISOINDOLE DERIVATIVES AS ANTIVIRAL DRUGS, AND NEW OXAZOLO 2,3-a]ISOINDOLE DERIVATIVES BOEHRINGER MANNHEIM GMBH (DE) 1995-10-11 EP disclosed