SCHEMBL9196802

SCHEMBL9196802

CC(C)c1cc(-c2ccccc2)cc(-c2ccc(F)cc2)c1S

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.39
TOP1 P11387 2/20 0.36
SQOR Q9Y6N5 1/20 0.35
USP1 O94782 1/20 0.34
WDR48 Q8TAF3 1/20 0.34
PTGS2 P35354 2/20 0.34
HPRT1 P00492 1/20 0.34
GCGR P47871 1/20 0.34
MAPK14 Q16539 1/20 0.34
STAT1 P42224 1/20 0.34
MEN1 O00255 1/20 0.33
FABP2 P12104 1/20 0.33
TSHR P16473 1/20 0.33
AKR1C4 P17516 1/20 0.33
ADRA2B P18089 1/20 0.33
CHRM3 P20309 1/20 0.33
PTGS1 P23219 1/20 0.33
HTR2C P28335 1/20 0.33
DRD3 P35462 1/20 0.33
AKR1C3 P42330 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9514015 0.94 HMGCR (0.42) HMGCRPTGS2GCGRPTGS1
SCHEMBL9514348 0.82 CA1 (0.47) HMGCRPTGS2MEN1FABP2TSHR
SCHEMBL24268972 0.80 CA1 (0.43) PTGS2
SCHEMBL9515012 0.80 HMGCR (0.44) HMGCRPTGS2GCGRPTGS1
SCHEMBL9857638 0.79 HMGCR (0.42) HMGCRGCGR
SCHEMBL9520263 0.78 HMGCR (0.39) HMGCRUSP1WDR48PTGS2HPRT1
SCHEMBL9857543 0.78 HMGCR (0.44) HMGCRPTGS2MEN1FABP2TSHR
SCHEMBL9512239 0.74 CA1 (0.53) HMGCRGCGRTSHRPTGS1HTR2C
SCHEMBL9512819 0.74 HMGCR (0.51) HMGCRKMT2A
SCHEMBL28968808 0.72 HMGCR (0.40) HMGCRPTGS2GCGRPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418648-B1 4-Hydroxytetrahydropyran-2-ones as well as the corresponding dehydroxy carbon acid derivatives, salts and esters, process for their preparation, pharmaceutical preparations as well as precursors HOECHST AG (DE) 1995-01-11 EP disclosed
US-5294724-A Anticholesterol agents HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-15 US disclosed
EP-0418648-A1 4-Hydroxytetrahydropyran-2-ones as well as the corresponding dehydroxy carbon acid derivatives, salts and esters, process for their preparation, pharmaceutical preparations as well as precursors HOECHST AKTIENGESELLSCHAFT (DE) 1991-03-27 EP disclosed